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1

Organic Reactions || The Barton-McCombie Reaction

McCombie, Stuart W.

Year:

2004

Language:

english

File:

PDF, 4.42 MB

english, 2004

2

Pyrroles and related compounds. Part XXIV. Separation and oxidative degradation of chlorophyll derivatives

Kenner, George W., McCombie, Stuart W., Smith, Kevin M.

Journal:

Journal of the Chemical Society Perkin Transactions 1

Year:

1973

Language:

english

File:

PDF, 943 KB

english, 1973

3

A novel method for the synthesis of aryl sulfones

Ruo W Steensma, Sharen Galabi, Jayaram R Tagat, Stuart W McCombie

Journal:

Tetrahedron Letters

Year:

2001

Language:

english

File:

PDF, 59 KB

english, 2001

4

Mild N-dealkylation of tertiary, benzylic amines with acid chlorides: Application to solid-phase chemistry

Michael W. Miller, Susan F. Vice, Stuart W. McCombie

Journal:

Tetrahedron Letters

Year:

1998

Language:

english

File:

PDF, 209 KB

english, 1998

5

A new method for the deoxygenation of secondary alcohols

Barton, Derek H. R., McCombie, Stuart W.

Journal:

Journal of the Chemical Society Perkin Transactions 1

Year:

1975

Language:

english

File:

PDF, 1.81 MB

english, 1975

6

Inhibition of the development of collagen-induced arthritis in rhesus monkeys by a small molecular weight antagonist of CCR5

Michel P. M. Vierboom, Paul J. Zavodny, Chuan-Chu Chou, Jayaram R. Tagat, Catherine Pugliese-Sivo, Julie Strizki, Ruo W. Steensma, Stuart W. McCombie, Liesbeth Çelebi-Paul, Ed Remarque, Margreet Jonke

Journal:

Arthritis & Rheumatism

Year:

2005

Language:

english

File:

PDF, 230 KB

english, 2005

7

ChemInform Abstract: New Reactions of Hydrazides. Part 1. Directed ortho- and Lateral Metalation of Aromatic Carbocyclic and Heterocyclic Systems.

Stuart W. McCombie, Sue-Ing Lin, Susan F. Vice

Journal:

Year:

2000

File:

PDF, 37 KB

2000

8

ChemInform Abstract: Suzuki Arylation of 1,1-Dibromo-1-alkenes: Synthesis of Tetra-Substituted Alkenes.

Annette Bauer, Michael W. Miller, Susan F. Vice, Stuart W. McCombie

Journal:

Year:

2001

File:

PDF, 30 KB

2001

9

ChemInform Abstract: A Novel Method for the Synthesis of Aryl Sulfones.

Ruo W. Steensma, Sharen Galabi, Jayaram R. Tagat, Stuart W. McCombie

Journal:

Year:

2001

File:

PDF, 27 KB

2001

10

ChemInform Abstract: Concise Formation of 4-Benzyl Piperidines and Related Derivatives Using a Suzuki Protocol.

Susan Vice, Stuart McCombie, et al. et al.

Journal:

Year:

2001

File:

PDF, 32 KB

2001

11

ChemInform Abstract: Piperazine-Based CCR5 Antagonists as HIV-1 Inhibitors. Part 1. 2(S)-Methyl Piperazine as a Key Pharmacophore Element.

Jayaram R. Tagat, Stuart W. McCombie, Ruo W. Steensma, Sue-Ing Lin, Dennis V. Nazareno, Bahige Baroudy, Nicole Vantuno, Serena Xu, Jia Liu

Journal:

Year:

2001

File:

PDF, 36 KB

2001

12

ChemInform Abstract: Synthesis and Structure—Activity Relationships of M2-Selective Muscarinic Receptor Ligands in the 1-[4-(4-Arylsulfonyl)phenylmethyl]-4-(4-piperidinyl)-piperazine Family.

Stuart W. McCombie, et al. et al.

Journal:

Year:

2002

File:

PDF, 31 KB

2002

13

ChemInform Abstract: Synthesis of Mono- and Difluoronaphthoic Acids.

Jayaram R. Tagat, Stuart W. McCombie, Dennis V. Nazareno, Craig D. Boyle, Joseph A. Kozlowski, Samuel Chackalamannil, Hubert Josien, Yuguang Wang, Guowei Zhou

Journal:

Year:

2002

File:

PDF, 31 KB

2002

14

Oximino-Piperidino-Piperidine-Based CCR5 Antagonists. Part 2. Synthesis, SAR and Biological Evaluation of Symmetrical Heteroaryl Carboxamides.

Anandan Palani, Sherry Shapiro, John W. Clader, William J. Greenlee, Susan Vice, Stuart McCombie, Kathleen Cox, Julie Strizki, Bahige M. Baroudy

Journal:

Year:

2003

File:

PDF, 171 KB

2003

15

Pyrrole und verwandte Verbindungen, XXI. Schutz der Porphyrinvinylgruppen. Eine Synthese von Koproporphyrin-III aus Protoporphyrin-IX2)

George W. Kenner, Stuart W. McCombie, Kevin M. Smith

Journal:

European Journal of Organic Chemistry

Year:

1973

File:

PDF, 636 KB

1973

16

Synthesis and in vitro activity of the penem antibiotics

Stuart W. McCombie, Ashit K. Ganguly

Journal:

Medicinal Research Reviews

Year:

1988

Language:

english

File:

PDF, 1.49 MB

english, 1988

17

A scalemic synthesis of the scopadulcic acid skeleton. II: Ring-D formation via regiospecific intramolecular aldol and alkylation reactions

Jayaram R. Tagat, Mohindar S. Puar, Stuart W. McCombie

Journal:

Tetrahedron Letters

Year:

1996

Language:

english

File:

PDF, 212 KB

english, 1996

18

A scalemic synthesis of the scopadulcic acid skeleton. I: An efficient γ-alkylation at C-9 in abietane framework and subsequent aldol reaction

Jayaram R. Tagat, Stuart W. McCombie, Mohindar S. Puar

Journal:

Tetrahedron Letters

Year:

1996

Language:

english

File:

PDF, 219 KB

english, 1996

19

Muscarinic M2 antagonists: anthranilamide derivatives with exceptional selectivity and in vivo activity

John W Clader, William Billard, Herbert Binch III, Lian-Yong Chen, Gordon Crosby Jr., Ruth A Duffy, Jennifer Ford, Joseph A Kozlowski, Jean E Lachowicz, Shengjian Li, Charles Liu, Stuart W McCombie, S

Journal:

Bioorganic & Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 240 KB

english, 2004

20

Synthetic inhibitors of interleukin-6 II: 3,5-diaryl pyridines and meta-terphenyls

Jayaram R. Tagat, Stuart W. McCombie, Beverly E. Barton, James Jackson, Jennifer Shortall

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 194 KB

english, 1995

21

Synthetic inhibitors of interleukin-6 I: 2,3,7,8-tetrahydro-4-aryl-1H-cyclopent [e] imidazo [1,2-a]- pyridin-5(6H)-one and related compounds

Jayaram R. Tagat, Dennis V. Nazareno, Stuart W. McCombie, Beverly E. Barton, Jennifer Shortall, James Jackson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 204 KB

english, 1995

22

Gamma-lactams and related compounds as cholesterol absorption inhibitors: homologs of the beta-lactam cholesterol absorption inhibitor SCH 484611

Sundeep Dugar, Michael P. Kirkup, John W. Clader, Sue-Ing Lin, Razia Rizvi, Mark E. Snow, Harry R. Davis Jr., Stuart W. McCombie

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 264 KB

english, 1995

23

(−)-SCH 57939: synthesis and pharmacological properties of a potent, metabolically stable cholesterol absorption inhibitor

Michael P. Kirkup, Razia Rizvi, Bandarpalle B. Shankar, Sundeep Dugar, John W. Clader, Stuart W. McCombie, Sue-Ing Lin, Nathan Yumibe, Keith Huie, Margaret Van Heek, Douglas S. Compton, Harry R. Davis

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 250 KB

english, 1996

24

Optimization of triaryl bis-sulfones as cannabinoid-2 receptor ligands

Brian J. Lavey, Joseph A. Kozlowski, Bandarpalle B. Shankar, James M. Spitler, Guowei Zhou, De-Yi Yang, Youheng Shu, Michael K.C. Wong, Shing-Chun Wong, Neng-Yang Shih, Jie Wu, Stuart W. McCombie, Raz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 166 KB

english, 2007

25

Non-aromatic A-ring replacement in the triaryl bis-sulfone CB2 receptor inhibitors

Eric J. Gilbert, Guowei Zhou, Michael K.C. Wong, Ling Tong, Bandarpalle B. Shankar, Chunli Huang, Joseph Kelly, Brian J. Lavey, Stuart W. McCombie, Lei Chen, Razia Rizvi, Youhao Dong, Youheng Shu, Jos

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 1.04 MB

english, 2010

26

Controlling benzylic functionality and stereochemistry: 2. Synthesis of the pseudopterosin aglycone

Stuart W. McCombie, Brian Cox, Ashit K. Ganduly

Journal:

Tetrahedron Letters

Year:

1991

Language:

english

File:

PDF, 273 KB

english, 1991

27

Controlling benzylic functionality and stereochemistry: 1. Synthesis of the secopseudopterosin aglycone

Stuart W. McCombie, Brian Cox, Sue-Ing Lin, Ashit K. Ganguly, Andrew T. McPhail

Journal:

Tetrahedron Letters

Year:

1991

Language:

english

File:

PDF, 255 KB

english, 1991

28

Synthesis of 3-heterosubstituted isocephem and iso-oxacephem antibiotics

Stuart W. McCombie, William A. Metz, Adriano Afonso

Journal:

Tetrahedron Letters

Year:

1986

Language:

english

File:

PDF, 211 KB

english, 1986

29

Cyclofunctionalisation of epoxyalcohol derivatives. 2. Stereo- and regiospecific conversion to 1,3-dioxolanes

Stuart W McCombie, William A Metz

Journal:

Tetrahedron Letters

Year:

1987

Language:

english

File:

PDF, 179 KB

english, 1987

30

Cyclofunctionalisation of epoxyalcohol derivatives. 1. Delivery of functionalised carbon for stereospecific synthesis of dihydrofurans and dihydroxyacids

Stuart W. McCombie, Bandarpalle B. Shankar, Ashit K. Ganguly

Journal:

Tetrahedron Letters

Year:

1985

Language:

english

File:

PDF, 194 KB

english, 1985

31

A concise route to the oxathiazepine containing eudistomin skeleton and some carba-analogs

Michael P. Kirkup, B.B. Shankar, Stuart McCombie, Ashit K. Ganguly, Andrew T. McPhail

Journal:

Tetrahedron Letters

Year:

1989

Language:

english

File:

PDF, 237 KB

english, 1989

32

Cyclofunctionalisation of epoxyalcohol derivatives. 4. Cyclisation of sulfonylacetate dianions: A synthesis of “MeBMT”

Stuart W. McCombie, Bandarpalle B. Shankar, Ashit K. Ganguly

Journal:

Tetrahedron Letters

Year:

1989

Language:

english

File:

PDF, 250 KB

english, 1989

33

One-pot, three-component synthesis of arylidenesuccinates and related compounds

Stuart W McCombie, Courtney A Luchaco

Journal:

Tetrahedron Letters

Year:

1997

Language:

english

File:

PDF, 117 KB

english, 1997

34

New reactions of hydrazides. Part 1: Directed ortho- and lateral metalation of aromatic carbocyclic and heterocyclic systems

Stuart W. McCombie, Sue-Ing Lin, Susan F. Vice

Journal:

Tetrahedron Letters

Year:

1999

Language:

english

File:

PDF, 248 KB

english, 1999

35

Indolocarbazoles. 1. Total synthesis and protein kinase inhibiting characteristics of compounds related to K-252c.

Stuart W McCombie, Robert W Bishop, Donna Carr, Emily Dobek, Michael P Kirkup, Paul Kirschmeier, Sue-Ing Lin, Joanne Petrin, Karen Rosinski, Bandarpalle B Shankar, Oswald Wilson

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1993

Language:

english

File:

PDF, 490 KB

english, 1993

36

Piperazine-Based CCR5 antagonists as HIV-1 inhibitors. I: 2(S)-methyl piperazine as a key pharmacophore element

Jayaram R. Tagat, Stuart W. McCombie, Ruo W. Steensma, Sue-Ing Lin, Dennis V. Nazareno, Bahige Baroudy, Nicole Vantuno, Serena Xu, Jia Liu

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 163 KB

english, 2001

37

Metabolic stabilization of benzylidene ketal M2 muscarinic receptor antagonists via halonaphthoic acid substitution

Craig D. Boyle, Samuel Chackalamannil, John W. Clader, William J. Greenlee, Hubert B. Josien, James J. Kaminski, Joseph A. Kozlowski, Stuart W. McCombie, Dennis V. Nazareno, Jayaram R. Tagat, Yuguang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 129 KB

english, 2001

38

Synthesis and anti-herpes activity of some a-ring functionalized dehydroabietane derivatives

Jayaram R. Tagat, Dennis V. Nazareno, Mohindar S. Puar, Stuart W. McCombie, Ashit K. Ganguly

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 324 KB

english, 1994

39

Indolocarbazole nitrogens linked by three-atom bridges: a potent new class of PKC inhibitors

Susan F. Vice, W.Robert Bishop, Stuart W. McCombie, Huong Dao, Emily Frank, Ashit K. Ganguly

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1994

Language:

english

File:

PDF, 494 KB

english, 1994

40

Synthesis and structure–Activity relationships of M2-Selective muscarinic receptor ligands in the 1-[4-(4-Arylsulfonyl)-phenylmethyl]-4-(4-piperidinyl)-piperazine family

Stuart W McCombie, Sue-Ing Lin, Jayaram R Tagat, Dennis Nazareno, Susan Vice, Jennifer Ford, Theodros Asberom, Daria Leone, Joseph A Kozlowski, Guowei Zhou, Vilma B Ruperto, Ruth A Duffy, Jean E Lacho

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 118 KB

english, 2002

41

Substituted 2-(R)-Methyl piperazines as muscarinic M2 selective ligands

Joseph A Kozlowski, Guowei Zhou, Jayaram R Tagat, Sue-Ing Lin, Stuart W McCombie, Vilma B Ruperto, Ruth A Duffy, Robert A McQuade, Gordon Crosby Jr., Lisa A Taylor, William Billard, Herbert Binch III,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 127 KB

english, 2002

42

Enhancement of pharmacokinetic properties and in vivo efficacy of benzylidene ketal M2 muscarinic receptor antagonists via benzamide modification

Craig D. Boyle, Susan F. Vice, Jennifer Campion, Samuel Chackalamannil, Claire M. Lankin, Stuart W. McCombie, William Billard, Herbert Binch, III, Gordon Crosby, Mary-Cohen Williams, Vicki L. Coffin,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 140 KB

english, 2002

43

Oximino-piperidino-piperidine-based CCR5 antagonists. Part 2: synthesis, SAR and biological evaluation of symmetrical heteroaryl carboxamides

Anandan Palani, Sherry Shapiro, John W. Clader, William J. Greenlee, Susan Vice, Stuart McCombie, Kathleen Cox, Julie Strizki, Bahige M. Baroudy

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 149 KB

english, 2003

44

Synthesis and chemistry of thia-analogs of the anti-mitotic podophyllium lignans

Stuart W. McCombie, Jayaram R. Tagat, William A. Metz, Dennis Nazareno, Mohindar S. Puar

Journal:

Year:

1993

Language:

english

File:

PDF, 1.03 MB

english, 1993

45

Synthesis of a C11 spiropiperidino derivative of 8-chloro-6,11-dihydro 5H-benzo[5,6]cyclohepta[1,2-b]pyridine

Adriano Afonso, J. Kelly, Mohindar S. Puar, Stuart McCombie, Andrew T. McPhail

Journal:

Tetrahedron Letters

Year:

1998

Language:

english

File:

PDF, 197 KB

english, 1998

46

Piperazine-based CCR5 antagonists as HIV-1 inhibitors. III: synthesis, antiviral and pharmacokinetic profiles of symmetrical heteroaryl carboxamides

Stuart W. McCombie, Jayaram R. Tagat, Susan F. Vice, Sue-Ing Lin, Ruo Steensma, Anandan Palani, Bernard R. Neustadt, Bahige M. Baroudy, Julie M. Strizki, Michael Endres, Kathleen Cox, Niya Dan, Chuan-

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2003

Language:

english

File:

PDF, 173 KB

english, 2003

47

Identification and characterization of pseudoirreversible nonpeptide antagonists of the neuropeptide Y Y5 receptor and development of a novel Y5-selective radioligand

Deborra Mullins, Nika Adham, David Hesk, Yusheng Wu, Joseph Kelly, Ying Huang, Mario Guzzi, Xiaoping Zhang, Stuart McCombie, Andrew Stamford, Eric Parker

Journal:

European Journal of Pharmacology

Year:

2008

Language:

english

File:

PDF, 807 KB

english, 2008

48

Interaction of small molecule inhibitors of HIV-1 entry with CCR5

Christoph Seibert, Weiwen Ying, Svetlana Gavrilov, Fotini Tsamis, Shawn E. Kuhmann, Anandan Palani, Jayaram R. Tagat, John W. Clader, Stuart W. McCombie, Bahige M. Baroudy, Steven O. Smith, Tatjana Dr

Journal:

Year:

2006

Language:

english

File:

PDF, 495 KB

english, 2006

49

Generation and in situ acylation of enaminone anions: a convenient synthesis of 3-carbethoxy-4(1H)-pyridinones and -4-pyrones and related compounds

McCombie, Stuart W., Metz, William A., Nazareno, Dennis, Shankar, Bandarpalle B., Tagat, Jayaram

Journal:

Journal of Organic Chemistry

Year:

1991

Language:

english

File:

PDF, 692 KB

english, 1991

50

Homogeneous, palladium(0)-catalyzed exchange deprotection of allylic esters, carbonates and carbamates

Jeffrey, Paul D., McCombie, Stuart W.

Journal:

Journal of Organic Chemistry

Year:

1982

Language:

english

File:

PDF, 610 KB

english, 1982